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| THURSDAY, MAY
9, 2002 |
| 08:30 - 09:20 |
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| PLENARY SESSION 4: BRZIN LECTURE |
| Chairperson: |
E. Reiner, Croatia |
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| 08:30 |
ACETYLCHOLINESTERASE
REGULATION IN SKELETAL MUSCLES
J. Sketelj, N. Crne-Finderle, P. Pregelj, Slovenia |
| 09:20 - 10:40 |
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| SESSION 14 |
| Chairperson: |
U. Drews, Germany |
|
| 09:20 |
CHOLINERGIC
CORTICAL TERMINATIONS ESTABLISH CLASSICAL SYNAPSES AND UNDERGO AGE-RELATED
ATROPHY
A.C. Cuello, P. Turrini, M.A. Casu, T.P. Wong, Y. De Koninck,
A. Ribeiro Da Silva, Canada |
| 09:40 |
DEVELOPMENT
OF CHOLINERGIC PROJECTIONS TO CORTEX: POSSIBLE ROLE OF NEUROTROPHINS
IN TARGET SELECTION
R. Robertson, J. Yu, USA |
| 10:00 |
ACTIVATION
OF THE CHOLINERGIC SYSTEM DURING COGNITIVE PROCESSES
G. Pepeu, M.G Giovannini, M. Pazzagli, J. Cangioli, M.B.
Passani, Italy |
| 10:20 |
PRECLINICAL
AND CLINICAL STUDIES ON THE ROLE OF MUSCARINIC RECEPTORS IN THE
PHARMACOTHERAPY OF SCHIZOPHRENIA
F.P. Bymaster, A. Shekhar, K.W. Perry, K. Rasmussen, D. McKinzie,
C.C. Felder, USA |
| 10:40 |
Coffee Break and Poster
Viewing |
| 11:10 - 12:50 |
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| SESSION 15 |
| Chairperson: |
K. Loffelholz, Germany |
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| 11:10 |
CENTRAL
CHOLINERGIC NEURONS IN CULTURE: REGULATION OF SURVIVAL AND FUNCTION
M. Segal, N. Landman, V. Greenberger, Israel |
| 11:30 |
HOW
IS THE BRAIN SUPPLIED WITH CHOLINE, BUT PROTECTED AGAINST EXCESS
CHOLINE?
K. Loffelholz, J. Klein, Germany |
| 11:50 |
MEASURING
CEREBRAL ACETYLCHOLINE ESTERASE ACTIVITY IN ALZHEIMER DEMENTIA BY
PET FUNCTIONAL PARAMETRIC IMAGING
K. Herholz, G. Zundorf, B. Bauer, S. Weisenbach, W-D. Heiss,
Germany |
| 12:10 |
BLOOD-BRAIN
BARRIER DISTRUPTION IS ASSOCIATED WITH ABNORMAL CORTICAL THETA RHYTHM
GENERATION: THE POTENTIAL INVOLVEMENT OF ACETYLCHOLINESTERASE
E. Aviv, I. Shelef, H. Golan, A. Korn, O. Tomkins, L. Pavlovsky,
A. Friedman, Israel |
| 12:30 |
CONTROL OF ACETYLCHOLINE
RELEASE UNDER STIMULATORY CONDITIONS BY ITS BIOSYNTHETIC PRECURSORS;
GLUCOSE AND CHOLINE
J. Klein, S. Kopf, K. Loeffelholz, Germany |
| 12:50 |
Lunch Break and Poster
Viewing |
| 14:45 - 16:25 |
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| SESSION 16 |
| Chairperson: |
A. Enz, Switzerland |
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| 14:45 |
TREATMENT
OF DEMENTIA WITH CHOLINESTERASE INHIBITORS
A.D. Korczyn, Israel |
| 15:05 |
CHOLINESTERASE
INHIBITORS STABILIZE COGNITIVE DECLINE IN ALZHEIMER'S DISEASE
E. Giacobini, Switzerland |
| 15:25 |
GENDER
DIFFERENCES IN THE ACTIONS OF CHOLINESTERASE INHIBITORS
M. Weinstock, R-H. Wang, Israel |
| 15:45 |
AMYLOID
PRECURSOR PROTEIN PROCESSING PROPERTIES OF THE NOVEL NEUROPROTECTIVE
CHOLINESTERASE MONOAMINE OXIDASE INHIBITOR,TV3326 AND ITS OPTICAL
ISOMER,TV3279
M.B.H. Youdim, M. Phalach-Yogev, O. Bar-Am, M. Weinstock,
T. Amit, Israel |
| 16:05 |
NOVEL
BIFUNCTIONAL COMPOUNDS ELICITING CHOLINERGIC AND ANTI-INFLAMMATORY
ACTIVITY FOR THE TREATMENT OF CNS IMPAIRMENTS
G. Amitai, R. Adani, I. Rabinovitz, G. Sod-Moriah, H. Meshulam,
Israel |
| 16:25 |
Coffee Break and Poster
Viewing |
| 17:00 - 18:20 |
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| SESSION 17 |
| Chairperson: |
S. Tucek, Czech Republic |
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| 17:00 |
ROLES
OF EXTERNAL LOOPS OF MUSCARINIC RECEPTORS IN INTERACTIONS BETWEEN
N-METHYLSCOPOLAMINE AND ALLOSTERIC MODULATORS
A. Krejci, S. Tucek, Czech Republic |
| 17:20 |
STRUCTURE
AND ACTIVATION OF MUSCARINIC ACETYLCHOLINE RECEPTORS
E.C. Hulme, Z-L. Lu, M.S. Bee, C.A.M. Curtis, UK |
| 17:40 |
GENERATION
AND ANALYSIS OF MUSCARINIC ACETYLCHOLINE RECEPTOR KNOCKOUT MICE
A. Duttaroy, M. Yamada, J. Gomeza, W. Zhang, R. Makita, T. Miyakawa,
F. Bymaster, C. Felder, C. Deng, J. Wess, USA, Japan |
| 18:00 |
CLOSING REMARKS
A.G. Karczmar, USA |
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